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Ryuta Yamazaki Selected Research

YHO-13351

4/2013ABCG2 inhibitor YHO-13351 sensitizes cancer stem/initiating-like side population cells to irinotecan.
7/2011Novel acrylonitrile derivatives, YHO-13177 and YHO-13351, reverse BCRP/ABCG2-mediated drug resistance in vitro and in vivo.

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Ryuta Yamazaki Research Topics

Disease

6Neoplasms (Cancer)
01/2021 - 12/2010
3Carcinoma (Carcinomatosis)
01/2021 - 10/2002
3Rheumatoid Arthritis
12/2002 - 07/2002
2Hematologic Neoplasms (Hematological Malignancy)
01/2021 - 01/2017
2Breast Neoplasms (Breast Cancer)
04/2013 - 07/2011
2Colonic Neoplasms (Colon Cancer)
07/2011 - 11/2002
2Inflammation (Inflammations)
01/2008 - 02/2004
1Pancreatic Neoplasms (Pancreatic Cancer)
07/2011
1Leukemia
07/2011
1Leukemia P388
07/2011
1Lung Neoplasms (Lung Cancer)
07/2011
1Hyperplasia
01/2008
1Alzheimer Disease (Alzheimer's Disease)
08/2005
1Stomach Neoplasms (Stomach Cancer)
08/2005
1Testicular Neoplasms (Testicular Cancer)
10/2002

Drug/Important Bio-Agent (IBA)

5Proteins (Proteins, Gene)FDA Link
05/2017 - 08/2005
3Irinotecan (Camptosar)FDA LinkGeneric
04/2013 - 10/2002
2proto-oncogene proteins pimIBA
01/2021 - 01/2017
2Transcription Factors (Transcription Factor)IBA
05/2017 - 12/2010
2YHO-13351IBA
04/2013 - 07/2011
2ProdrugsIBA
07/2011 - 10/2002
2Prostaglandin-Endoperoxide Synthases (Cyclooxygenase)IBA
01/2008 - 11/2002
2Cyclooxygenase 2 Inhibitors (COX-2 Inhibitors)IBA
01/2008 - 11/2002
2Non-Steroidal Anti-Inflammatory Agents (NSAIDs)IBA
01/2008 - 07/2002
1ThiazolidinedionesIBA
01/2021
1Phosphotransferases (Kinase)IBA
01/2021
1methanesulfonic acid (methanesulfonate)IBA
01/2021
1Serine (L-Serine)FDA Link
01/2017
1Antineoplastic Agents (Antineoplastics)IBA
01/2017
1Threonine (L-Threonine)FDA Link
01/2017
1Member 1 Subfamily B ATP Binding Cassette TransporterIBA
07/2011
1Paclitaxel (Taxol)FDA LinkGeneric
07/2011
1Topotecan (Hycamtin)FDA LinkGeneric
07/2011
1Doxorubicin (Adriamycin)FDA LinkGeneric
07/2011
1YHO-13177IBA
07/2011
1Mitoxantrone (Novantrone)FDA LinkGeneric
07/2011
1Pharmaceutical PreparationsIBA
12/2010
1Celecoxib (Celebrex)FDA Link
01/2008
1Presenilin-2IBA
08/2005
1CalciumIBA
08/2005
1Carrier Proteins (Binding Protein)IBA
08/2005
1Cycloheximide (Cicloheximide)IBA
08/2005
1Fluorouracil (Carac)FDA LinkGeneric
08/2005
1InterferonsIBA
08/2005
1IntegrinsIBA
08/2005
1triptolideIBA
02/2004
1Sodium Salicylate (Salicylate, Sodium)IBA
12/2002
1Aspirin (Acetylsalicylic Acid)FDA LinkGeneric
12/2002
1Cyclooxygenase 2 (Cyclooxygenase-2)IBA
12/2002
1Anti-Inflammatory Agents (Anti-Inflammatories)IBA
12/2002
1Etoposide (VP 16)FDA LinkGeneric
10/2002
1Cisplatin (Platino)FDA LinkGeneric
10/2002
1BromidesIBA
10/2002
1PPAR gammaIBA
07/2002

Therapy/Procedure

2Drug Therapy (Chemotherapy)
04/2013 - 07/2011
1Therapeutics
05/2017